Molecule Details
InChIKeyZSBBASZUYKREPU-PRHODGIISA-N
Canonical SMILESCc1c(-c2ccc(Br)cc2)nsc1NC(=O)[C@@H]1C[C@H]1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13255 GRM1 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 8.2 IC50 ChEMBL;BindingDB
P41594 GRM5 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 6.1 IC50 ChEMBL;BindingDB