Molecule Details
InChIKeyZRZMENVDJBJBOY-HOCLYGCPSA-N
Compound Name6-(6-cyclopropylimidazo[1,2-a]pyridin-3-yl)-N-((3R,4S)-4-(trifluoromethyl)pyrrolidin-3-yl)pyridin-2-amine
Canonical SMILESFC(F)(F)[C@H]1CNC[C@@H]1Nc1cccc(-c2cnc3ccc(C4CC4)cn23)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.38
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 9.2 IC50 BindingDB
Q9NWZ3 IRAK4 Homo sapiens Human PF07714 9.2 IC50 BindingDB
P51617 IRAK1 Homo sapiens Human PF00531 PF00069 6.7 IC50 BindingDB