Molecule Details
InChIKeyZRMHSSFCCBYNHY-ZDUSSCGKSA-N
Compound Name[4-[2-(methylamino)-2-oxoethoxy]phenyl]methyl (2S)-2-[(4-sulfamoylphenyl)carbamothioylamino]propanoate
Canonical SMILESCNC(=O)COc1ccc(COC(=O)[C@H](C)/N=C(\S)Nc2ccc(S(N)(=O)=O)cc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.8 Ki ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.8 pIC50 TTD_MultiTarget
P00915 CA1 Homo sapiens Human PF00194 7.2 Ki ChEMBL;BindingDB