Molecule Details
InChIKeyZRKHDIABAALLSW-WSDLNYQXSA-N
Compound NameN,2-dimethyl-5-nitro-N-[(E)-(5-pyridin-3-ylpyrazolo[1,5-a]pyrimidin-3-yl)methylideneamino]benzenesulfonamide
Canonical SMILESCc1ccc([N+](=O)[O-])cc1S(=O)(=O)N(C)/N=C/c1cnn2ccc(-c3cccnc3)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.16
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 8.1 IC50 ChEMBL;BindingDB
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 6.7 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 6.7 IC50 ChEMBL