Molecule Details
InChIKeyZRAYFKGWJMRLBX-UHFFFAOYSA-N
Compound Name2-[5-Fluoro-6-(1-oxo-2,3-dihydroisoindol-5-yl)-1,3-benzothiazole-2-carbonyl]-5-[(sulfamoylamino)methyl]-1,3,4-oxadiazole
Canonical SMILESNS(=O)(=O)NCc1nnc(C(=O)c2nc3cc(F)c(-c4ccc5c(c4)CNC5=O)cc3s2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y5X9 LIPG Homo sapiens Human PF00151 PF01477 8.3 IC50 ChEMBL;BindingDB
P11150 LIPC Homo sapiens Human PF00151 PF01477 7.7 IC50 ChEMBL;BindingDB