Molecule Details
InChIKeyZQTAUZWIZMXKIL-UHFFFAOYSA-N
Compound NameN-cyclopropyl-4-oxo-1-[3-[4-[2-(2H-tetrazol-5-yl)cyclopropyl]phenyl]phenyl]-1,8-naphthyridine-3-carboxamide
Canonical SMILESO=C(NC1CC1)c1cn(-c2cccc(-c3ccc(C4CC4c4nnn[nH]4)cc3)c2)c2ncccc2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.26
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27815 PDE4A Homo sapiens Human PF18100 PF00233 9.3 IC50 ChEMBL;BindingDB
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 9.3 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 9.3 IC50 ChEMBL;BindingDB