Molecule Details
InChIKeyZQLILUVVXPRXLE-UHFFFAOYSA-N
Compound Name6-Acetyl-8-cyclopentyl-5-methyl-2-[[5-(4-prop-2-enoylpiperazin-1-yl)-2-pyridinyl]amino]pyrido[2,3-d]pyrimidin-7-one
Canonical SMILESC=CC(=O)N1CCN(c2ccc(Nc3ncc4c(C)c(C(C)=O)c(=O)n(C5CCCC5)c4n3)nc2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.17
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00534 CDK6 Homo sapiens Human PF00069 7.8 IC50 ChEMBL
P11802 CDK4 Homo sapiens Human PF00069 7.6 IC50 ChEMBL
Q9NYV4 CDK12 Homo sapiens Human PF00069 6.0 IC50 ChEMBL