Molecule Details
InChIKeyZQIKAKSHLZASKW-UHFFFAOYSA-N
Compound Nametert-butyl 2-(N-(6-cyano-1-((1-methyl-1H-imidazol-5-yl)methyl)-1,2,3,4-tetrahydroquinolin-3-yl)pyridine-2-sulfonamido)acetate
Canonical SMILESCn1cncc1CN1CC(N(CC(=O)OC(C)(C)C)S(=O)(=O)c2ccccn2)Cc2cc(C#N)ccc21
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.82
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.8 IC50 ChEMBL