Molecule Details
InChIKeyZQEBKQUIKOLFRO-UHFFFAOYSA-N
Compound Name1-(4-Fluorophenyl)-4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazine
Canonical SMILESFc1ccc(N2CCN(Cc3cnn(-c4ccccc4)c3)CC2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P21917 DRD4 Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB