Molecule Details
InChIKeyZPKLGSLFCKFOCY-UHFFFAOYSA-N
Compound NameN-[3-[6-amino-5-(3,4,5-trimethoxyphenyl)-3-pyridinyl]phenyl]methanesulfonamide
Canonical SMILESCOc1cc(-c2cc(-c3cccc(NS(C)(=O)=O)c3)cnc2N)cc(OC)c1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q04771 ACVR1 Homo sapiens Human PF01064 PF07714 PF08515 8.2 IC50 ChEMBL;BindingDB
P36897 TGFBR1 Homo sapiens Human PF01064 PF00069 PF08515 6.7 IC50 ChEMBL;BindingDB
P06241 FYN Homo sapiens Human PF07714 PF00017 PF00018 6.3 IC50 ChEMBL;BindingDB