Molecule Details
InChIKeyZPHPMNJCCXXCGX-UHFFFAOYSA-N
Compound Name4-[3-(3-Amino-phenyl)-1-hydroxy-1-(3-methyl-3H-imidazol-4-yl)-prop-2-ynyl]-2-naphthalen-1-yl-benzonitrile
Canonical SMILESCn1cncc1C(O)(C#Cc1cccc(N)c1)c1ccc(C#N)c(-c2cccc3ccccc23)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.45
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.2 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.2 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 7.0 IC50 ChEMBL;BindingDB