Molecule Details
InChIKeyZPHNUQZFJFUCHA-UHFFFAOYSA-N
Compound Name2-amino-4-[4-(azetidin-3-ylsulfonyl)-3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl]-1,3-benzothiazole-7-carboxylic acid
Canonical SMILESNc1nc2c(-c3ccc(S(=O)(=O)C4CNC4)c(S(N)(=O)=O)c3-c3nn[nH]n3)ccc(C(=O)O)c2s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.97
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.5 IC50 ChEMBL;BindingDB
P52699 Serratia marcescens Pathogen PF00753 9.9 IC50 BindingDB
Q9XAY4 blaVIM Pseudomonas aeruginosa Pathogen PF00753 9.5 IC50 BindingDB