Molecule Details
InChIKeyZOZPVKJSFYNWLP-VMPREFPWSA-N
Compound Name[(S)-1-[(S)-1-(4-Benzoyl-piperidine-1-carbonyl)-3-methyl-butylcarbamoyl]-2-(1H-indol-3-yl)-ethyl]-carbamic acid tert-butyl ester
Canonical SMILESCC(C)C[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)OC(C)(C)C)C(=O)N1CCC(C(=O)c2ccccc2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.04
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.0 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB