Molecule Details
InChIKeyZOWREHOVFWKKPQ-UHFFFAOYSA-N
Compound Name2-[(1-Aminoisoquinolin-6-yl)amino]-7-tert-butylsulfonyl-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(19),6,8,10(21),16(20),17-hexaene-3,12-dione
Canonical SMILESCC(C)(C)S(=O)(=O)c1ccc2cc1CNC(=O)C(Nc1ccc3c(N)nccc3c1)c1ccc(cc1)CCCC(=O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06870 KLK1 Homo sapiens Human PF00089 7.7 Ki ChEMBL;BindingDB
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 7.5 Ki ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 7.5 Ki ChEMBL