Molecule Details
InChIKeyZOJCSVHWXFCTBG-UHFFFAOYSA-N
Compound Name3-[2-[4-(3,4-Dichlorophenyl)piperazin-1-yl]ethyl]-1,5-dimethylpyrimido[5,4-b]indole-2,4-dione
Canonical SMILESCn1c(=O)n(CCN2CCN(c3ccc(Cl)c(Cl)c3)CC2)c(=O)c2c1c1ccccc1n2C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.44
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB