Molecule Details
InChIKeyZOHXHAYMXURWLP-MNNMKWMVSA-N
Compound Name(6S,7S)-5-acetyl-N-hydroxy-6-(4-phenyl-3,4-dihydro-2H-pyridine-1-carbonyl)-5-azaspiro[2.5]octane-7-carboxamide
Canonical SMILESCC(=O)N1CC2(CC2)C[C@H](C(=O)NO)[C@H]1C(=O)N1C=CC(c2ccccc2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.12
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.3 pIC50 TTD_MultiTarget
O14672 ADAM10 Homo sapiens Human PF21299 PF00200 PF13574 7.3 IC50 ChEMBL;BindingDB
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 6.8 IC50 ChEMBL;BindingDB