Molecule Details
InChIKeyZOBKJVAECISXJA-UHFFFAOYSA-N
Canonical SMILESCOc1cc(Nc2nccc(Oc3ccc(NC(=O)Nc4cc(C5CC5)nn4-c4ccc(C)cc4)c4ccccc34)n2)cc(C(=O)NCCN2CCOCC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.1
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
P43405 SYK Homo sapiens Human PF07714 PF00017 7.5 IC50 ChEMBL;BindingDB