Molecule Details
InChIKeyZMXFWVYPMCRPSG-UHFFFAOYSA-N
Compound NameN-[2-methoxy-4-(1-methylpiperidin-4-yl)oxyphenyl]-3-propan-2-yl-2,5,11,13-tetrazatricyclo[7.4.0.02,6]trideca-1(13),3,5,7,9,11-hexaen-12-amine
Canonical SMILESCOc1cc(OC2CCN(C)CC2)ccc1Nc1ncc2ccc3ncc(C(C)C)n3c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.12
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P24385 CCND1 Homo sapiens Human PF02984 PF00134 7.1 IC50 ChEMBL;BindingDB
Q00534 CDK6 Homo sapiens Human PF00069 7.1 IC50 ChEMBL