Molecule Details
InChIKeyZMIXZDFAIQPNIS-UHFFFAOYSA-N
Compound Name4-[4-(Cyclohexylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidine
Canonical SMILESc1c(N2CCCC2)nc(N2CCCC2)nc1N1CCN(CC2CCCCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29466 CASP1 Homo sapiens Human PF00619 PF00656 7.3 IC50 ChEMBL;BindingDB
P51878 CASP5 Homo sapiens Human PF00619 PF00656 6.9 IC50 ChEMBL;BindingDB
P49662 CASP4 Homo sapiens Human PF00619 PF00656 6.3 IC50 ChEMBL;BindingDB