Molecule Details
InChIKeyZMHJLQHDDUQJEC-UWUNEBHHSA-N
Canonical SMILESCOc1ccc(F)cc1-c1c(F)cnc2[nH]c(C3CCN([C@H]4CC[C@@H](CC(=O)O)CC4)CC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 7.4 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 7.4 IC50 ChEMBL