Molecule Details
InChIKeyZKVURPUQVABYSC-UHFFFAOYSA-N
Compound Name4-(4-chlorophenyl)-1-cyclopropyl-3-ethyl-5-(8-methoxy-3-methyl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)-4H-pyrrolo[3,4-d]pyrazol-6-one
Canonical SMILESCCc1nn(C2CC2)c2c1C(c1ccc(Cl)cc1)N(c1cc(OC)c3nnc(C)n3c1)C2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60885 BRD4 Homo sapiens Human PF17035 PF17105 PF00439 7.5 IC50 ChEMBL;BindingDB
P25440 BRD2 Homo sapiens Human PF17035 PF00439 7.4 IC50 ChEMBL;BindingDB
Q15059 BRD3 Homo sapiens Human PF17035 PF00439 7.2 IC50 ChEMBL;BindingDB