Molecule Details
InChIKeyZKNQRQDTAWUUJL-UHFFFAOYSA-N
Compound Name2-[4-[4-(4-Methyl-3,5-dioxo-1,2,4-triazin-2-yl)butyl]piperazin-1-yl]benzonitrile
Canonical SMILESCn1c(=O)cnn(CCCCN2CCN(c3ccccc3C#N)CC2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)4
Pfam Stratification Homologous
Avg pChEMBL8.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (4)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.1 Ki ChEMBL
P35348 ADRA1A Homo sapiens Human PF00001 8.1 Ki ChEMBL
P35368 ADRA1B Homo sapiens Human PF00001 8.1 Ki ChEMBL