Molecule Details
InChIKeyZKNCPHDOHBCAIF-CYBMUJFWSA-N
Compound Name8-(3-Methylimidazo[l,2-a]pyridin-6-yl)-7-(oxazo l-2-yl)-2-((tetrahydrofiiran-3-yl)methyl)-[l,2,4] triazolo[l,5-c]pyrimidin-5-amine (isomer 2)
Canonical SMILESCc1cnc2ccc(-c3c(-c4ncco4)nc(N)n4nc(C[C@H]5CCOC5)nc34)cn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 9.3 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB