Molecule Details
InChIKeyZKDTULNFGWCQJA-UHFFFAOYSA-N
Compound Name1-[4-(2,3-Dihydro-benzo[1,4]dioxin-5-yl)-piperazin-1-yl]-2-[8-(4-methyl-piperazin-1-yl)-naphthalen-2-yloxy]-ethanone
Canonical SMILESCN1CCN(c2cccc3ccc(OCC(=O)N4CCN(c5cccc6c5OCCO6)CC4)cc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28222 HTR1B Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB