Molecule Details
InChIKeyZJOQXNGTEXFLLO-UHFFFAOYSA-N
Compound NameN,6-dihydroxy-2-(4-methoxyphenyl)sulfonyl-3,4-dihydro-1H-isoquinoline-1-carboxamide
Canonical SMILESCOc1ccc(S(=O)(=O)N2CCc3cc(O)ccc3C2C(=O)NO)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.17
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P51511 MMP15 Homo sapiens Human PF11857 PF00045 PF00413 PF01471 6.2 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 6.1 pIC50 TTD_MultiTarget