Molecule Details
InChIKeyZIOWEXJTMJYIOK-UHFFFAOYSA-N
Compound NameN-[1-(5,5-dimethyl-2,4-dioxoimidazolidin-1-yl)-3-[4-[4-(trifluoromethoxy)phenyl]phenoxy]propan-2-yl]-N-hydroxyformamide
Canonical SMILESCC1(C)C(=O)NC(=O)N1CC(COc1ccc(-c2ccc(OC(F)(F)F)cc2)cc1)N(O)C=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.68
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.4 pIC50 TTD_MultiTarget
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 7.7 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 6.9 IC50 ChEMBL;BindingDB