Molecule Details
InChIKeyZIJYBRHNQICJRS-WVGFPPCDSA-N
Compound Name[(1S,2S,3R,11S,12S,14R,15R,18R,20S)-18-(2-fluorophenyl)-3-hydroxy-1,11,15-trimethyl-5-oxo-7-pyridin-3-yl-6,10,17,19-tetraoxapentacyclo[12.8.0.02,11.04,9.015,20]docosa-4(9),7-dien-12-yl] 4-cyanobenzoate
Canonical SMILESC[C@@]12CO[C@@H](c3ccccc3F)O[C@H]1CC[C@@]1(C)[C@H]2C[C@H](OC(=O)c2ccc(C#N)cc2)[C@@]2(C)Oc3cc(-c4cccnc4)oc(=O)c3[C@H](O)[C@H]12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O75908 SOAT2 Homo sapiens Human PF03062 8.2 IC50 ChEMBL;BindingDB
P35610 SOAT1 Homo sapiens Human PF03062 6.5 IC50 ChEMBL;BindingDB