Molecule Details
InChIKeyZIATUPKJNZVSLT-UHFFFAOYSA-N
Compound NameCyclohexyl-[6-piperazin-1-yl-4-(2H-pyrazol-3-yl)[2,4'']bipyridinyl-2''-yl]amine
Canonical SMILESc1cc(-c2cc(-c3cc[nH]n3)cc(N3CCNCC3)n2)cc(NC2CCCCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.61
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15139 PRKD1 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 8.4 IC50 ChEMBL;BindingDB
Q13563 PKD2 Homo sapiens Human PF18109 PF08016 PF20519 7.2 IC50 BindingDB
Q9BZL6 PRKD2 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 7.2 IC50 ChEMBL