Molecule Details
InChIKeyZHZRYPWKMPTDMQ-SANMLTNESA-N
Compound Name(2S)-N-[4-[3-cyano-1-(2-methyl-1-oxo-3H-isoindol-5-yl)indol-5-yl]oxyphenyl]pyrrolidine-2-carboxamide
Canonical SMILESCN1Cc2cc(-n3cc(C#N)c4cc(Oc5ccc(NC(=O)[C@@H]6CCCN6)cc5)ccc43)ccc2C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16875 PFKFB3 Homo sapiens Human PF01591 PF00300 7.5 IC50 ChEMBL;BindingDB
O60825 PFKFB2 Homo sapiens Human PF01591 PF00300 7.0 IC50 ChEMBL;BindingDB
P16118 PFKFB1 Homo sapiens Human PF01591 PF00300 6.2 IC50 ChEMBL;BindingDB