Molecule Details
InChIKeyZHTQHERQPPHQPE-UJGSWJOCSA-N
Compound NameDes-AA1,2,5-[D-Agl8(NbetaMe,2-naphthoyl),IAmp9, m-I-Tyr11]SRIF
Canonical SMILESCC(C)NCc1ccc(C[C@@H]2NC(=O)[C@H](N(C)C(=O)c3ccc4ccccc4c3)NC(=O)[C@H](Cc3ccccc3)NC(=O)[C@@H](Cc3ccccc3)NC(=O)[C@@H](CCCCN)NC(=O)[C@H](N)CSSC[C@@H](C(=O)O)NC(=O)[C@H](CO)NC(=O)[C@@H]([C@@H](C)O)NC(=O)[C@H](Cc3ccc(O)cc3I)NC(=O)[C@@H]([C@@H](C)O)NC2=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.93
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30872 SSTR1 Homo sapiens Human PF00001 8.2 IC50 ChEMBL;BindingDB
P31391 SSTR4 Homo sapiens Human PF00001 6.4 IC50 ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 6.3 IC50 ChEMBL;BindingDB