Molecule Details
InChIKeyZHSFCHXKHOJYIG-SFHVURJKSA-N
Canonical SMILESCC[C@H](NS(=O)(=O)c1ccc(-c2sc(-c3nnc(CC(C)(C)C(=O)O)o3)nc2CC2CCCCC2)c(C(F)F)c1F)C(F)(F)F
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.23
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P51449 RORC Homo sapiens Human PF00104 PF00105 8.4 IC50 ChEMBL;BindingDB
Q92753 RORB Homo sapiens Human PF00104 PF00105 6.0 IC50 ChEMBL;BindingDB