Molecule Details
InChIKeyZGULUKQLEOFSEK-UHFFFAOYSA-N
Compound Name2-((1H-pyrrolo[2,3-b]pyridin-5-yl)oxy)-4-(1-((6-(4-chlorophenyl)spiro[3.5]non-6-en-7-yl)methyl)-1,2,3,6-tetrahydropyridin-4-yl)-N-((3-nitro-4-(((tetrahydro-2H-pyran-4-yl)methyl)amino)phenyl)sulfonyl)benzamide
Canonical SMILESO=C(NS(=O)(=O)c1ccc(NCC2CCOCC2)c([N+](=O)[O-])c1)c1ccc(C2=CCN(CC3=C(c4ccc(Cl)cc4)CC4(CCC4)CC3)CC2)cc1Oc1cnc2[nH]ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.21
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10415 BCL2 Homo sapiens Human PF00452 PF02180 8.6 IC50 ChEMBL;BindingDB
O43521 BCL2L11 Homo sapiens Human PF08945 PF06773 8.2 IC50 BindingDB
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 7.8 IC50 BindingDB