Molecule Details
InChIKeyZGQHZEDUFBEHQX-UHFFFAOYSA-N
Compound Name4-[9-[4-(benzenesulfonamido)phenyl]-3,3,6,6-tetramethyl-1,8-dioxo-4,5,7,9-tetrahydro-2H-acridin-10-yl]benzenesulfonamide
Canonical SMILESCC1(C)CC(=O)C2=C(C1)N(c1ccc(S(N)(=O)=O)cc1)C1=C(C(=O)CC(C)(C)C1)C2c1ccc(NS(=O)(=O)c2ccccc2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00918 CA2 Homo sapiens Human PF00194 7.0 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 6.2 Ki ChEMBL;BindingDB
O43570 CA12 Homo sapiens Human PF00194 6.2 Ki ChEMBL;BindingDB