Molecule Details
InChIKeyZFTPEIAEGCLUII-WYLSNLDWSA-M
Compound Namep-Tyr(SO3Na)-gNle-mGly-Trp-(N-Me)Nle-Asp-Phe-NH2
Canonical SMILESCCCC[C@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CNC(=O)[C@H](CCCC)NC(=O)[C@@H](N)Cc1ccc(OS(=O)(=O)[O-])cc1)C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccccc1)C(N)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL10.22
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 10.2 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 10.2 Ki ChEMBL;BindingDB