Molecule Details
InChIKeyZFOPWBXSJXQVFA-UHFFFAOYSA-N
Compound NameN-(4-morpholin-4-ylsulfonylphenyl)-3-(1H-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amine
Canonical SMILESO=S(=O)(c1ccc(Nc2nccn3c(-c4cn[nH]c4)cnc23)cc1)N1CCOCC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.1 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB