Molecule Details
InChIKeyZDZWIYNKACEWQC-UHFFFAOYSA-N
Compound Name5-cyano-N-[2-(cyclohexen-1-yl)-4-[1-[2-(1H-imidazol-5-yl)acetyl]piperidin-4-yl]phenyl]-1H-imidazole-2-carboxamide
Canonical SMILESN#Cc1c[nH]c(C(=O)Nc2ccc(C3CCN(C(=O)Cc4c[nH]cn4)CC3)cc2C2=CCCCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.18
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07333 CSF1R Homo sapiens Human PF00047 PF25305 PF07714 9.0 IC50 ChEMBL;BindingDB
P11712 CYP2C9 Homo sapiens Human PF00067 6.5 IC50 ChEMBL;BindingDB
P33261 CYP2C19 Homo sapiens Human PF00067 6.1 IC50 ChEMBL;BindingDB