Molecule Details
InChIKeyZDSWMSRFTNIEJV-UHFFFAOYSA-N
Compound Name7-(3-(trifluoromethyl)pyridin-2-yl)-N-(5-(trifluoromethyl)pyridin-2-yl)-1,8-naphthyridin-4-amine
Canonical SMILESFC(F)(F)c1ccc(Nc2ccnc3nc(-c4ncccc4C(F)(F)F)ccc23)nc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.33
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q8NER1 TRPV1 Homo sapiens Human PF00023 PF12796 PF00520 8.7 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB