Molecule Details
InChIKeyZDRGLSBALZDWBH-MPEHDAKKSA-N
Compound Name(13S)-17-(tert-butylcarbamoyl)-13-methyl-6,7,8,9,11,12,14,15-octahydrocyclopenta[a]phenanthrene-3-carboxylic acid
Canonical SMILESCC(C)(C)NC(=O)C1=CCC2C3CCc4cc(C(=O)O)ccc4C3CC[C@]12C
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.22
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 7.2 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 7.2 pIC50 TTD_MultiTarget