Molecule Details
InChIKeyZDBWMZVBCYVNPS-FIFLTTCUSA-N
Compound NameN-hydroxy-3-(1-methyl-4-(3-oxo-3-phenylprop-1-enyl)-1H-pyrrol-2-yl)acrylamide
Canonical SMILESCn1cc(/C=C/C(=O)c2ccccc2)cc1/C=C/C(=O)NO
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.59
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 6.6 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.6 pIC50 TTD_MultiTarget
Q92769 HDAC2 Homo sapiens Human PF00850 6.6 pIC50 TTD_MultiTarget