Molecule Details
InChIKeyZDASUJMDVPTNTF-UHFFFAOYSA-N
Canonical SMILESOc1c(Br)cc(Br)c2cccnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.04
SourceBindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB13536
Drug NameBroxyquinoline
CAS Number521-74-4
Groups experimental
ATC Codes P01AA01 A07AX01 G01AC06
Descriptionnan

Categories: Alimentary Tract and Metabolism Antidiarrheals, Intestinal Antiinflammatory/antiinfective Agents Antiparasitic Products, Insecticides and Repellents Antiprotozoals Genito Urinary System and Sex Hormones Gynecological Antiinfectives and Antiseptics Heterocyclic Compounds, Fused-Ring Hydroxyquinoline Derivatives Hydroxyquinolines Intestinal Antiinfectives Quinoline Derivatives Quinolines
Cross-references: BindingDB: 76301 ChEBI: 109543 CHEMBL223448 ChemSpider: 2359 Wikipedia: Broxyquinoline ZINC: ZINC000000001064
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 6.0 Ki BindingDB
Q9K2N0 blaVIM-2 Pseudomonas aeruginosa Pathogen PF00753 6.0 Ki BindingDB