Molecule Details
InChIKeyZCZSJYUQIMCWOG-FCSANXPSSA-N
Canonical SMILESCOc1ccc(CC[C@@H](OC(=O)[C@@H]2CCCCN2C(=O)[C@H](c2cc(OC)c(OC)c(OC)c2)c2ccc(C)s2)c2cccc(OCCN3CCOCC3)c2)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.55
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13451 FKBP5 Homo sapiens Human PF00254 PF00515 PF13181 7.0 IC50 ChEMBL
Q02790 FKBP4 Homo sapiens Human PF00254 PF00515 PF07719 6.1 Ki ChEMBL