Molecule Details
InChIKeyZCRJVXDJCMBFCS-UHFFFAOYSA-N
Compound Name1-{5-oxo-1H,2H,3H,5H,9bH-benzo[a]pyrrolizin-9-yl}-3-[5-(pyrrolidin-1-ylmethyl)-1H-pyrazol-3-yl]urea
Canonical SMILESO=C(Nc1cc(CN2CCCC2)[nH]n1)Nc1cccc2c1C1CCCN1C2=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.33
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 6.3 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.3 pIC50 TTD_MultiTarget