Molecule Details
InChIKeyZCNHSWBTKSJQNS-UHFFFAOYSA-N
Compound Name1-[[3-[[4-(4-Methylpiperazin-1-yl)-3-(trifluoromethyl)benzoyl]amino]phenyl]methylamino]phthalazine-5-carboxamide
Canonical SMILESCN1CCN(c2ccc(C(=O)Nc3cccc(CNc4nncc5c(C(N)=O)cccc45)c3)cc2C(F)(F)F)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
Q96GD4 AURKB Homo sapiens Human PF00069 8.2 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 7.2 IC50 ChEMBL;BindingDB