Molecule Details
InChIKeyZCLCUGHPNSTPGZ-FQEVSTJZSA-N
Compound Name(R)-4-Dipentylcarbamoyl-4-[(1H-indole-2-carbonyl)-amino]-butyric acid
Canonical SMILESCCCCCN(CCCCC)C(=O)[C@H](CCC(=O)O)NC(=O)c1cc2ccccc2[nH]1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.77
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 6.8 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 6.8 IC50 ChEMBL;BindingDB