Molecule Details
InChIKeyZBLLHXCRPWKVCY-UHFFFAOYSA-N
Compound Name4-(Cyclohexylamino)-6-piperazin-1-yl-1,3,5-triazine-2-carbonitrile
Canonical SMILESN#Cc1nc(NC2CCCCC2)nc(N2CCNCC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.36
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 9.0 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.8 IC50 ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 6.3 IC50 ChEMBL;BindingDB