Molecule Details
InChIKeyZAZVLBZIEZHJFV-BEFAXECRSA-N
Compound Name(S)-7-(5-fluoro-2-methylbenzyloxy)-2-((R)-2-methylpiperazin-1-yl)-6,7-dihydro-5H-cyclopenta[b]pyridine
Canonical SMILESCc1ccc(F)cc1CO[C@H]1CCc2ccc(N3CCNC[C@H]3C)nc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.98
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28335 HTR2C Homo sapiens Human PF00001 8.8 IC50 ChEMBL;BindingDB
P41595 HTR2B Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 7.3 IC50 ChEMBL;BindingDB