Molecule Details
InChIKeyZAZPPOBRQFIKRC-UHFFFAOYSA-N
Compound Name6-fluoro-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4-dihydroisoquinolin-1(2H)-one
Canonical SMILESCOc1ccccc1N1CCN(CCCCN2CCc3cc(F)ccc3C2=O)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.6 Ki ChEMBL
P14416 DRD2 Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB