Molecule Details
InChIKeyZANNOGKZSUYAAD-UHFFFAOYSA-N
Compound NamePyrazolo[1,5-b]pyridazine deriv. 53
Canonical SMILESCOc1cc(Nc2nccc(-c3cnn4nc(C)ccc34)n2)cc(C(F)(F)F)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.8
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 7.7 pIC50 TTD_MultiTarget