Molecule Details
InChIKeyZAKSQHPNZWUBFJ-UHFFFAOYSA-N
Canonical SMILESCOc1cn(C(CCOC(C)(C)C)C(=O)Nc2ccc3nn(C)cc3c2)c(=O)cc1-c1cc(Cl)ccc1-n1cc(Cl)nn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.59
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P03951 F11 Homo sapiens Human PF00024 PF00089 8.8 IC50 ChEMBL;BindingDB
P03952 KLKB1 Homo sapiens Human PF00024 PF00089 8.4 IC50 ChEMBL;BindingDB