Molecule Details
InChIKeyZAIFESHMEUUZQE-OAHLLOKOSA-N
Compound Name2-[[(2R)-1-methylpyrrolidin-2-yl]methyl]-4-pentylphthalazin-1-one
Canonical SMILESCCCCCc1nn(C[C@H]2CCCN2C)c(=O)c2ccccc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.03
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35367 HRH1 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35348 ADRA1A Homo sapiens Human PF00001 6.3 pIC50 TTD_MultiTarget
P35368 ADRA1B Homo sapiens Human PF00001 6.0 Ki ChEMBL